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Structure-Based Design of a Chemical Probe Set for the 5‑HT5A Serotonin Receptor.

• Authors : Levit Kaplan, Anat; Strachan, Ryan T.; Braz, Joao M.

• Source: Journal of Medicinal Chemistry; 3/10/2022, Vol. 65 Issue 5, p4201-4217, 17p

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Polyazamacrocycle Ligands Facilitate 89Zr Radiochemistry and Yield 89Zr Complexes with Remarkable Stability.

• Authors : Pandya, Darpan N.; Henry, Kelly E.; Day, Cynthia S.

• Source: Inorganic Chemistry; 12/7/2020, Vol. 59 Issue 23, p17473-17487, 15p

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The Peculiar Trend of Cyclic Perfluoroalkane Electron Affinities with Increasing Ring Size.

• Authors : Paul, Ankan¹; Wannere, Chaitanya S.¹; Kasalova, Veronica¹

Subjects: *ATOMIC orbitals; *ELECTRONS; *FUNCTIONAL analysis

• Source: Journal of the American Chemical Society. 11/9/2005, Vol. 127 Issue 44, p15457-15469. 13p.

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Structure-Based Design of a Chemical Probe Set for the 5-HT 5A Serotonin Receptor.

• Authors : Levit Kaplan A; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, California 94143, United States.; Strachan RT

Subjects: Serotonin* ; Serotonin Antagonists*/Serotonin Antagonists*/Serotonin Antagonists*/pharmacology; Humans

• Source: Journal of medicinal chemistry [J Med Chem] 2022 Mar 10; Vol. 65 (5), pp. 4201-4217. Date of Electronic Publication: 2022 Feb 23.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic

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Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y 14 R Antagonist.

• Authors : Wen Z; Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892, United States.; Salmaso V

Subjects: Piperidines/Piperidines/Piperidines/*chemistry ; Purinergic P2 Receptor Antagonists/Purinergic P2 Receptor Antagonists/Purinergic P2 Receptor Antagonists/*pharmacology; Animals

• Source: Journal of medicinal chemistry [J Med Chem] 2022 Feb 24; Vol. 65 (4), pp. 3434-3459. Date of Electronic Publication: 2022 Feb 03.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic

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Structure-Activity Relationship of Heterocyclic P2Y 14 Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres.

• Authors : Jung YH; Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892, United States.; Salmaso V

Subjects: Piperidines/Piperidines/Piperidines/*chemistry ; Purinergic P2 Receptor Antagonists/Purinergic P2 Receptor Antagonists/Purinergic P2 Receptor Antagonists/*chemistry ; Receptors, Purinergic P2/Receptors, Purinergic P2/Receptors, Purinergic P2/*metabolism

• Source: Journal of medicinal chemistry [J Med Chem] 2021 Apr 22; Vol. 64 (8), pp. 5099-5122. Date of Electronic Publication: 2021 Mar 31.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic

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Polyazamacrocycle Ligands Facilitate 89 Zr Radiochemistry and Yield 89 Zr Complexes with Remarkable Stability.

• Authors : Pandya DN; Department of Radiology, University of Iowa, Iowa City, Iowa 52242, United States.; Henry KE

• Source: Inorganic chemistry [Inorg Chem] 2020 Dec 07; Vol. 59 (23), pp. 17473-17487. Date of Electronic Publication: 2020 Nov 10.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0366543 Publication Model: Print-Electronic

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Exploration of Alternative Scaffolds for P2Y 14 Receptor Antagonists Containing a Biaryl Core.

• Authors : Jung YH; Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892, United States.; Yu J

Subjects: Drug Design*; Purinergic P2 Receptor Antagonists/Purinergic P2 Receptor Antagonists/Purinergic P2 Receptor Antagonists/*chemistry ; Purinergic P2 Receptor Antagonists/Purinergic P2 Receptor Antagonists/Purinergic P2 Receptor Antagonists/*pharmacology

• Source: Journal of medicinal chemistry [J Med Chem] 2020 Sep 10; Vol. 63 (17), pp. 9563-9589. Date of Electronic Publication: 2020 Aug 06.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic

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Synthetic Antimicrobial Peptide Tuning Permits Membrane Disruption and Interpeptide Synergy.

• Authors : Fields FR; Department of Biology, University of Notre Dame, Notre Dame, Indiana 46556, United States.; Eck Institute of Global Health, University of Notre Dame, Notre Dame, Indiana 46556, United States.

• Source: ACS pharmacology & translational science [ACS Pharmacol Transl Sci] 2020 Feb 21; Vol. 3 (3), pp. 418-424. Date of Electronic Publication: 2020 Feb 21 (Print Publication: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101721411 Publication Model: eCollection

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